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Litlhaloso tsa Ethylmethyl-Carbamic Chloride;N-Ethyl-N-Methylcarbamoyl Chloride

Litlhaloso tsa Ethylmethyl-Carbamic Chloride;N-Ethyl-N-Methylcarbamoyl Chloride

Tlhaloso e Khutšoanyane:

CAS no: 42252-34-6

Lintho tsa lik'hemik'hale: Rivastigmine tartrate Intermediates


Lintlha tsa Sehlahisoa

Li-tag tsa Sehlahisoa

Etsa mosebetsi o felletseng oa ho khotsofatsa litlhoko tsohle tsa bareki ba rona;fumana lintlafatso tse tsoelang pele ka ho khothaletsa nts'etsopele ea bareki ba rona;hola ho ba molekane oa ho qetela oa tšebelisano-'moho le bareki le ho holisa lithahasello tsa bareki bakeng sa Quots bakeng sa Ethylmethyl-Carbamic Chloride;N-Ethyl-N-Methylcarbamoyl Chloride, esale re batla ho theha mekhatlo ea litšebelisano 'moho le uena.Etsa bonnete ba hore u ikopanya le rona bakeng sa lintlha tse ling.
Etsa mosebetsi o felletseng oa ho khotsofatsa litlhoko tsohle tsa bareki ba rona;fumana lintlafatso tse tsoelang pele ka ho khothaletsa nts'etsopele ea bareki ba rona;hola ho ba molekane oa ho qetela oa tšebelisano 'moho oa bareki le ho holisa lithahasello tsa bareki bakeng saChina Ethylmethyl-Carbamic Chloride;N-Ethyl-N-, Re bile molekane oa hau ea tšepahalang limmarakeng tsa machaba tsa lintho tsa rona.Re tsepamisitse maikutlo ho faneng ka litšebeletso ho bareki ba rona e le ntho ea bohlokoa ho matlafatsa likamano tsa rona tsa nako e telele.Ho lula ho le teng ha lihlahisoa tsa boemo bo holimo hammoho le tšebeletso ea rona e ntle ea pele le ka mor'a thekiso ho netefatsa tlholisano e matla 'marakeng o ntseng o eketseha oa lefatše.Re ikemiselitse ho sebelisana le metsoalle ea khoebo e tsoang hae le kantle ho naha, ho theha bokamoso bo botle.Rea u amohela ho Etela feme ea rona.Re lebeletse ho ba le tšebelisano-'moho le uena.

Ethylmethyl-carbamic chloride e sebelisoa e le karolo e bohareng ea Rivastigmine tartrate.
Rivastigmine tartrate ke rivastigmine lefu la Alzheimer lithethefatsi, rivastigmine ke physostigmine derivative ke Novartis ka lekhetlo la pele ka katleho ntshetswa pele lebitso la khoebo Exelon (exelon), molek'hule le moo carbamate sebopeho, ke mofuta oa amino acid ea selective cerebral cholinesterase inhibitor, e ka boela ea thibela. the acetylcholinesterase le butyrylcholinesterase, cholinergic neurons ka ho liehisa ho lokolloa ha acetylcholine degradation le matla a khothalletsang cholinergic nerve conduction, e ka ntlafatsa mathata a ts'ebetso ea kelello a kenngoeng ke cholinergic, kahoo e ntlafatsa ts'ebetso ea kelello ea bakuli ba lefu la Alzheimer's.Rivastigmine plasma e tlamang protheine e fokola, habonolo ka mokoallo oa mali-boko, o nang le tekanyo e phahameng ea khetho ea boko.Ha e khetholle feela hore e sebetsa ho cerebral cortex le hippocampus e amehang habonolo, empa hape e thibela ka mokhoa o ikhethileng mofuta o ka sehloohong oa AChE bokong, e leng se bakang phokotso ea katleho ea litla-morao tsa peripheral cholinergic.Rivastigmine in vivo halofo ea bophelo ke nako e khuts'oane le e telele ea ketso.Ho fapana le tacrine, sehlahisoa sena se hippocampus le cortex ea G1 enzyme inhibitory effect se matla.Tleliniki bakeng sa kalafo ea 'dementia' e bobebe ho isa ho e itekanetseng ea mofuta oa Alzheimer, kapa lefu la Alzheimer's ho ka belaelloa hore ke lefu la Alzheimer's Clinical.

Etsa mosebetsi o felletseng oa ho khotsofatsa litlhoko tsohle tsa bareki ba rona;fumana lintlafatso tse tsoelang pele ka ho khothaletsa nts'etsopele ea bareki ba rona;hola ho ba molekane oa ho qetela oa tšebelisano-'moho le bareki le ho holisa lithahasello tsa bareki bakeng sa Quots bakeng sa Ethylmethyl-Carbamic Chloride;N-Ethyl-N-Methylcarbamoyl Chloride, esale re batla ho theha mekhatlo ea litšebelisano 'moho le uena.Etsa bonnete ba hore u ikopanya le rona bakeng sa lintlha tse ling.
Quots bakeng saChina Ethylmethyl-Carbamic Chloride;N-Ethyl-N-, Re bile molekane oa hau ea tšepahalang limmarakeng tsa machaba tsa lintho tsa rona.Re tsepamisitse maikutlo ho faneng ka litšebeletso ho bareki ba rona e le ntho ea bohlokoa ho matlafatsa likamano tsa rona tsa nako e telele.Ho lula ho le teng ha lihlahisoa tsa boemo bo holimo hammoho le tšebeletso ea rona e ntle ea pele le ka mor'a thekiso ho netefatsa tlholisano e matla 'marakeng o ntseng o eketseha oa lefatše.Re ikemiselitse ho sebelisana le metsoalle ea khoebo e tsoang hae le kantle ho naha, ho theha bokamoso bo botle.Rea u amohela ho Etela feme ea rona.Re lebeletse ho ba le tšebelisano-'moho le uena.


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